发明名称 Polymorphs of acyl sulfonamides
摘要 The application discloses novel polymorphic crystalline forms of 2-[4-Bromo-3-(3-chloro-5-cyano-phenoxy)-2-fluoro-phenyl]-N-(2-chloro-4-propionylsulfamoyl-phenyl)-acetamide, sodium salt (Ib) with improved stability and physical properties which facilitate manufacturing, handling and formulating for treatment or prophylaxis of HIV mediated diseases, AIDS or ARC, in monotherapy or in combination therapy.
申请公布号 US8063103(B2) 申请公布日期 2011.11.22
申请号 US20090556235 申请日期 2009.09.09
申请人 DAVIDSON JAMES PRENTICE;PANG FEI;WONG MARGARET;MARTIN MICHAEL;ROCHE PALO ALTO LLC 发明人 DAVIDSON JAMES PRENTICE;PANG FEI;WONG MARGARET;MARTIN MICHAEL
分类号 C07C311/51;A61K31/277 主分类号 C07C311/51
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