发明名称 INHIBITORS OF PROTEIN TYROSINE KINASE ACTIVITY AND USE THEREOF TO TREAT OPHTHALMIC DISORDERS
摘要 Disclosed are compounds, and compositions of same, that are protein tyrosine kinase inhibitors. The compounds find use in the treatment of ophthalmic diseases, disorders and conditions. Said compounds are of the formulae (I), (II) or (III). Wherein R = (IV), (V), (VI), (VII), (VIII), (IX), (X), (XI) or (XII).
申请公布号 CA2796054(A1) 申请公布日期 2011.10.20
申请号 CA20112796054 申请日期 2011.04.08
申请人 METHYLGENE INC. 发明人 CLARIDGE, STEPHEN WILLIAM;GAUDETTE, FREDERIC;RAEPPEL, FRANCK;RAEPPEL, STEPHANE;VAISBURG, ARKADII;ZHAN, LIJIE
分类号 C07D495/04;A61K31/4365;A61K31/444;A61K31/496;A61K31/5377;A61P27/02 主分类号 C07D495/04
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