发明名称 HETEROARYL SUBSTITUTED PYRROLO[2,3-B]PYRIDINES AND PYRROLO[2,3-B]PYRIMIDINES AS JANUS KINASE INHIBITORS
摘要 The present invention provides heteroaryl substituted pyrrolo[2,3-b]pyridines (I) and heteroaryl substituted pyrrolo[2,3-b]pyrimidines that modulate the activity of Janus kinases and are useful in the treatment of diseases related to activity of Janus kinases including, for example, immune-related diseases, skin disorders, myeloid proliferative disorders, cancer, and other diseases.
申请公布号 EP1966202(B1) 申请公布日期 2011.09.21
申请号 EP20060839328 申请日期 2006.12.12
申请人 INCYTE CORPORATION 发明人 RODGERS, JAMES D.;SHEPARD, STACEY;MADUSKUIE, THOMAS P.;WANG, HAISHENG;FALAHATPISHEH, NIKOO;RAFALSKI, MARIA;ARVANITIS, ARGYRIOS G.;STORACE, LOUIS;JALLURI, RAVI KUMAR;FRIDMAN, JORDAN S.;VADDI, KRISHNA
分类号 C07D471/04;A61K31/395;A61P17/00;A61P35/00;A61P37/00;C07D487/04 主分类号 C07D471/04
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