发明名称 |
HETEROARYL SUBSTITUTED PYRROLO[2,3-B]PYRIDINES AND PYRROLO[2,3-B]PYRIMIDINES AS JANUS KINASE INHIBITORS |
摘要 |
The present invention provides heteroaryl substituted pyrrolo[2,3-b]pyridines (I) and heteroaryl substituted pyrrolo[2,3-b]pyrimidines that modulate the activity of Janus kinases and are useful in the treatment of diseases related to activity of Janus kinases including, for example, immune-related diseases, skin disorders, myeloid proliferative disorders, cancer, and other diseases. |
申请公布号 |
EP1966202(B1) |
申请公布日期 |
2011.09.21 |
申请号 |
EP20060839328 |
申请日期 |
2006.12.12 |
申请人 |
INCYTE CORPORATION |
发明人 |
RODGERS, JAMES D.;SHEPARD, STACEY;MADUSKUIE, THOMAS P.;WANG, HAISHENG;FALAHATPISHEH, NIKOO;RAFALSKI, MARIA;ARVANITIS, ARGYRIOS G.;STORACE, LOUIS;JALLURI, RAVI KUMAR;FRIDMAN, JORDAN S.;VADDI, KRISHNA |
分类号 |
C07D471/04;A61K31/395;A61P17/00;A61P35/00;A61P37/00;C07D487/04 |
主分类号 |
C07D471/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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