| 发明名称 |
N-(3-phenylamino-quinoxalin-2-yl)-benzenesulfonamide derivatives as phosphatidylinositol 3-kinase inhibitors |
| 摘要 |
The present invention comprises small molecule inhibitors of phosphatidylinositol 3-kinase (PI3K), which is associated with a number of malignancies such as ovarian cancer, cervical cancer, breast cancer, colon cancer, rectal cancer, and gioblastomas, among others. Accordingly, the compounds of the present invention are useful for treating, preventing, and/or inhibiting these diseases. |
| 申请公布号 |
EP2364974(A1) |
申请公布日期 |
2011.09.14 |
| 申请号 |
EP20110167227 |
申请日期 |
2006.10.09 |
| 申请人 |
EXELIXIS, INC. |
发明人 |
BAJJALIEH, WILLIAM;BANNEN, LYNNE, CANNE;BROWN, S., DAVID;KEARNEY, PATRICK;MAC, MORRISON;MARLOWE, CHARLES, K.;NUSS, JOHN, M.;TESFAI, ZEROM;WANG, YONG;XU, WEI |
| 分类号 |
C07D241/44;A61K31/498;A61K31/4985;A61P35/00;C07D401/12;C07D403/12;C07D405/12;C07D407/12;C07D409/12;C07D413/12;C07D417/12 |
主分类号 |
C07D241/44 |
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