发明名称 PROCESS FOR THE PREPARATION OF 1- ( 3-HYDROXYMETHYLPYRID-2 -YL ) -2 -PHENYL-4-METHYLPIPERAZINE AND MIRTAZAPINE
摘要 Disclosed herein is a process for the manufacture of mirtazapine and intermediates useful in preparing mirtazapine which includes the reduction of 1-(3-carboxypyridyl-2)-4-methyl-2-phenylpiperazine with an organoaluminum hydride.
申请公布号 US2011201804(A1) 申请公布日期 2011.08.18
申请号 US200913063085 申请日期 2009.10.20
申请人 WATSON PHARMA PRIVATE LIMITED 发明人 BHANU MANJUNATH NARAYAN;NAIK SAMIR;JOSHI PRASHANT;SHARMA VIJAY
分类号 C07D487/14;C07D401/04 主分类号 C07D487/14
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