发明名称 ONE-STEP PROCESS FOR PREPARING PALIPERIDONE AND ITS OXALATE SALT.
摘要 <p>The present invention relates to a one-step process for the preparation of the antipsychotic agent Paliperidone by oxidation of Risperidone, and to Paliperidone oxalate or a hydrate, solvate or polymorph thereof.</p>
申请公布号 MX2011006715(A) 申请公布日期 2011.07.20
申请号 MX20110006715 申请日期 2009.12.15
申请人 CHEMO IBERICA, S.A. 发明人 CASTALDI, GRAZIANO;RASPARINI, MARCELLO;MARRAS, GIOVANNI;BANFI, LUCA;DE MOLINER, FABIO;MUSUMECI, FRANCESCA;RIVA, RENATA
分类号 C07D471/04;A61K31/517;A61P25/00 主分类号 C07D471/04
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