发明名称 |
ONE-STEP PROCESS FOR PREPARING PALIPERIDONE AND ITS OXALATE SALT. |
摘要 |
<p>The present invention relates to a one-step process for the preparation of the antipsychotic agent Paliperidone by oxidation of Risperidone, and to Paliperidone oxalate or a hydrate, solvate or polymorph thereof.</p> |
申请公布号 |
MX2011006715(A) |
申请公布日期 |
2011.07.20 |
申请号 |
MX20110006715 |
申请日期 |
2009.12.15 |
申请人 |
CHEMO IBERICA, S.A. |
发明人 |
CASTALDI, GRAZIANO;RASPARINI, MARCELLO;MARRAS, GIOVANNI;BANFI, LUCA;DE MOLINER, FABIO;MUSUMECI, FRANCESCA;RIVA, RENATA |
分类号 |
C07D471/04;A61K31/517;A61P25/00 |
主分类号 |
C07D471/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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