发明名称 Salts of {1-methyl-5-[2-(5-trifluoromethyl-1H-imidazol-2-yl)-pyridin-4-yloxy]-1H-benzoimidazol-2-yl}-(4-trifluromethyl-phenyl)amine
摘要 Disclosed is a salt of {1-methyl-5-[2-(5-trifluoromethyl-1H-imidazol-2-yl)-pyridin-4-yloxy]-1H-benzoimidazol-2-yl}-(4-trifluoromethyl-phenyl)amine selected from the group consisting of acetate, tosylate, succinate, lactate, malate, sulfate, maleate, citrate, hydrochloride, phosphate, ethanesulfonate, and methanesulfonate, or a solvate and/or hydrate thereof. The salt is useful for treating cancer and inhibiting angiogenesis.
申请公布号 NZ574620(A) 申请公布日期 2011.05.27
申请号 NZ20070574620 申请日期 2007.08.30
申请人 NOVARTIS AG 发明人 GULLAPALLI, RAMPURNA;HASHASH, AHMAD;KARPINSKI, PIOTR, H;LIN, KANGWEN, L;LOESER, ERIC, M;OKHAMAFE, AUGUSTUS, O;SUTTON, PAUL, ALLEN;SY, EDUARDO
分类号 C07D401/14;A61K31/4439;A61P35/00 主分类号 C07D401/14
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