发明名称 |
Salts of {1-methyl-5-[2-(5-trifluoromethyl-1H-imidazol-2-yl)-pyridin-4-yloxy]-1H-benzoimidazol-2-yl}-(4-trifluromethyl-phenyl)amine |
摘要 |
Disclosed is a salt of {1-methyl-5-[2-(5-trifluoromethyl-1H-imidazol-2-yl)-pyridin-4-yloxy]-1H-benzoimidazol-2-yl}-(4-trifluoromethyl-phenyl)amine selected from the group consisting of acetate, tosylate, succinate, lactate, malate, sulfate, maleate, citrate, hydrochloride, phosphate, ethanesulfonate, and methanesulfonate, or a solvate and/or hydrate thereof. The salt is useful for treating cancer and inhibiting angiogenesis.
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申请公布号 |
NZ574620(A) |
申请公布日期 |
2011.05.27 |
申请号 |
NZ20070574620 |
申请日期 |
2007.08.30 |
申请人 |
NOVARTIS AG |
发明人 |
GULLAPALLI, RAMPURNA;HASHASH, AHMAD;KARPINSKI, PIOTR, H;LIN, KANGWEN, L;LOESER, ERIC, M;OKHAMAFE, AUGUSTUS, O;SUTTON, PAUL, ALLEN;SY, EDUARDO |
分类号 |
C07D401/14;A61K31/4439;A61P35/00 |
主分类号 |
C07D401/14 |
代理机构 |
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