发明名称 DERIVATIVES OF 5-AMINO-4,6-DISUBSTITUTED INDOLE AND 5-AMINO-4,6-DISUBSTITUTED INDOLINE AS POTASSIUM CHANNEL MODULATORS
摘要 This invention provides compounds of formula I where the dashed line represents an optional double bond; where R1 is phenyl, naphthyl, pyridyl, pyrimidyl, pyrrolyl, imidazolyl, pyrazyl, furyl, thienyl, oxazolyl, isoxazolyl, thiazolyl, or isothiazolyl, optionally substituted, and other substituents are defined herein. Such compounds are potassium channel modulators.
申请公布号 US2011118318(A1) 申请公布日期 2011.05.19
申请号 US20100856514 申请日期 2010.08.13
申请人 VALEANT PHARMACEUTICALS INTERNATIONAL 发明人 VERNIER JEAN-MICHEL;CHEN HUANMING;SONG JIANLAN
分类号 A61K31/4439;A61K31/404;C07D209/22;C07D401/06 主分类号 A61K31/4439
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