发明名称 |
CARVEDILOL PHOSPHATE SALT AND/OR SOLVATE THEREOF, CORRESPONDING COMPOSITION, AND/OR METHOD OF TREATMENT |
摘要 |
PROBLEM TO BE SOLVED: To provide a composition for treatment of hypertension, congestive heart failure and angina. SOLUTION: There are provided a carvedilol phosphate salt containing a crystal form of carvedilol dihydrogen phosphate (i.e., dihydrogen phosphate salt of 1-(carbazol-4-yloxy-3-[[2-(o-methoxyphenoxy)ethyl]amino]-2-propanol) and/or carvedilol hydrogen phosphate, etc.) having high water solubility, chemical stability, etc., and/or its solvate, and a composition containing the salt and/or the solvate. COPYRIGHT: (C)2011,JPO&INPIT
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申请公布号 |
JP2011088917(A) |
申请公布日期 |
2011.05.06 |
申请号 |
JP20100282048 |
申请日期 |
2010.12.17 |
申请人 |
SMITHKLINE BEECHAM (CORK) LTD |
发明人 |
BROOK CHRISTOPHER S;CHEN WEI;DELL'ORCO PHILIP C;KATRINCIC LEE M;LOUVET ANN MARIE;OH CHOON K;SPOORS PAUL G;WERNER CHRISTOPHER |
分类号 |
A61K31/403;C07D209/88;A61P9/00;A61P9/04;A61P9/10;A61P9/12;C07D209/82 |
主分类号 |
A61K31/403 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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