发明名称 Process for producing aminoacetyl pyrrolidine carbonitrile derivative and intermediate for production thereof
摘要 Novel intermediates for the production of aminoacetyl pyrrolidine carbonitrile derivatives ensure the safe and efficient production of the compounds. Specifically, the present invention provides a sulfonyloxyacetyl pyrrolidine derivative, represented by the following formula: (Chemical Formula 1) (wherein R1 is a substituted or unsubstituted C1-C6 alkyl group, a substituted or unsubstituted C3-C6 cycloalkyl group, a substituted or unsubstituted arylmethyl group, a substituted or unsubstituted aromatic hydrocarbon, a substituted or unsubstituted aromatic heterocyclic ring or a substituted or unsubstituted aliphatic heterocyclic ring; R2 is CONH2 or CN; and X is CH2, CHF or CF2.)
申请公布号 US7915427(B2) 申请公布日期 2011.03.29
申请号 US20070224849 申请日期 2007.02.02
申请人 KYORIN PHARMACEUTICALS CO., LTD. 发明人 ASAHINA YOSHIKAZU;FUKUDA YASUMICHI;SHIGA FUTOSHI
分类号 C07D207/04 主分类号 C07D207/04
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