发明名称 FORMULIERUNGEN VON BORSÄURE-VERBINDUNGEN
摘要 The present invention provides stable compounds prepared from boronic acid and lyophilized compounds thereof of formula (1) in which Z 1 and Z 2 are moieties derived from sugar. The invention also provides methods for preparing such compounds. Lyophilizing a mixture comprising a boronic acid compound and a moiety derived from sugar produces a stable composition that readily releases the boronic acid compound upon reconstitution in aqueous media.
申请公布号 AT501157(T) 申请公布日期 2011.03.15
申请号 AT20020709145T 申请日期 2002.01.25
申请人 THE UNITED STATES OF AMERICA, REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES 发明人 GUPTA, SHANKER
分类号 A61K9/19;C07F5/02;A61K31/69;A61K38/00;A61K38/05;A61K38/14;A61P29/00;A61P31/18;A61P35/00;A61P37/02;A61P43/00;C07F5/04;C07F5/05;C07H9/00;C07K5/06;C07K5/062;C07K5/065;C07K5/078;C07K5/08;C07K5/083;C07K5/097;C07K5/117;C07K7/02;C07K9/00 主分类号 A61K9/19
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