发明名称 |
FORMULIERUNGEN VON BORSÄURE-VERBINDUNGEN |
摘要 |
The present invention provides stable compounds prepared from boronic acid and lyophilized compounds thereof of formula (1) in which Z 1 and Z 2 are moieties derived from sugar. The invention also provides methods for preparing such compounds. Lyophilizing a mixture comprising a boronic acid compound and a moiety derived from sugar produces a stable composition that readily releases the boronic acid compound upon reconstitution in aqueous media. |
申请公布号 |
AT501157(T) |
申请公布日期 |
2011.03.15 |
申请号 |
AT20020709145T |
申请日期 |
2002.01.25 |
申请人 |
THE UNITED STATES OF AMERICA, REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES |
发明人 |
GUPTA, SHANKER |
分类号 |
A61K9/19;C07F5/02;A61K31/69;A61K38/00;A61K38/05;A61K38/14;A61P29/00;A61P31/18;A61P35/00;A61P37/02;A61P43/00;C07F5/04;C07F5/05;C07H9/00;C07K5/06;C07K5/062;C07K5/065;C07K5/078;C07K5/08;C07K5/083;C07K5/097;C07K5/117;C07K7/02;C07K9/00 |
主分类号 |
A61K9/19 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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