发明名称 SUBSTITUTED PIPERIDINE COMPOUNDS AND METHODS OF THEIR USE
摘要 Novel 3,4-disubstituted-4-aryl-piperidine compounds are disclosed. Pharmaceutical compositions containing the 3,4-disubstituted-4-aryl-piperidine compounds and methods of their pharmaceutical uses are also disclosed. The compounds disclosed are useful, inter alia, as antagonists of opioid receptors.
申请公布号 US2011034417(A1) 申请公布日期 2011.02.10
申请号 US20100897824 申请日期 2010.10.05
申请人 ADOLOR CORPORATION 发明人 LE BOURDONNEC BERTRAND;DOLLE ROLAND E.
分类号 A61K31/451;A61K31/435;A61K31/4468;A61K31/454;A61K31/4545;A61K31/4725;A61K31/485;A61K31/5377;A61K31/675;A61P1/00;A61P1/08;A61P1/10;A61P29/00;C07D211/22;C07D211/34;C07D401/06;C07D401/12;C07D413/12;C07F9/38;C07F9/59 主分类号 A61K31/451
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