发明名称 |
A NOVEL AND EFFICIENT METHOD FOR THE SYNTHESIS OF AN AMINO ACID |
摘要 |
<p>The present invention relates to a novel process for the preparation ofγ-amino acids, such as (±)-3-(aminomethyl)-5-methyl-hexanoic acid (1), which is a key intermediate in the preparation of the potent anticonvulsant pregabalin, (S)-(+)-3-(aminomethyl)-5-methyl-hexanoic acid (2), and its analogues.</p> |
申请公布号 |
EP2280930(A1) |
申请公布日期 |
2011.02.09 |
申请号 |
EP20090757806 |
申请日期 |
2009.06.03 |
申请人 |
GENERICS [UK] LIMITED;MYLAN DEVELOPMENT CENTRE PRIVATE LIMITED |
发明人 |
GORE, VINAYAK;GADAKAR, MAHESHKUMAR;SHINDE, DATTATREYA |
分类号 |
C07C227/04;A61K31/197;A61P25/00;C07C205/15;C07C205/51;C07C229/08 |
主分类号 |
C07C227/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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