发明名称 |
INDOLES AS MODULATORS OF NICOTICIC ACETYLCHOLINE RECEPTOR SUBTYPE ALPHA-7 |
摘要 |
The present invention relates to modulation of the α7 nicotinic acetylcholine receptor (nAChR) by a compound of List A or a salt thereof, which may be represented, but is not limited to the compound N-[(2-Trifluoromethyl-1H-indol-5-yl)methyl]-5-(trifluoromethyl)-2-pyrimidinecarboxamide.
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申请公布号 |
US2011028486(A1) |
申请公布日期 |
2011.02.03 |
申请号 |
US20090936431 |
申请日期 |
2009.04.16 |
申请人 |
DINNELL KEVIN;LIGHTFOOT ANDREW P;MARSHALL HOWARD ROBERT |
发明人 |
DINNELL KEVIN;LIGHTFOOT ANDREW P.;MARSHALL HOWARD ROBERT |
分类号 |
A61K31/501;A61K31/4155;A61K31/4196;A61K31/427;A61K31/4439;A61K31/444;A61K31/497;A61K31/506;A61P25/18;C07D401/12;C07D401/14;C07D403/12;C07D417/12 |
主分类号 |
A61K31/501 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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