发明名称 |
HETEROCYCLIC SULFONAMIDE INHIBITOR AGAINST BETA-AMYLOID PRODUCTION |
摘要 |
PROBLEM TO BE SOLVED: To provide compounds for inhibiting the production of aβ-amyloid protein from an amyloid precursor protein (APP), and to provide drugs used for treating Altzheimer's disease and Down's syndrome by using the compounds. SOLUTION: There are provided compounds represented by formula (I), pharmaceutically acceptable salts, hydrates and/or prodrugs thereof. COPYRIGHT: (C)2011,JPO&INPIT
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申请公布号 |
JP2010265280(A) |
申请公布日期 |
2010.11.25 |
申请号 |
JP20100144307 |
申请日期 |
2010.06.24 |
申请人 |
WYETH LLC;ARQULE INC |
发明人 |
KREFT ANTHONY FRANK;COLE DEREK CECIL;WOLLER KEVIN ROGER;STOCK JOSEPH RAYMOND;DIAMANITIS GEORGE;KURBRAK DENNIS MICHAEL;KUTTERER KRISTINA MARTHA;MOORE WILLIAM JAY;CASEBIER DAVID SCOTT |
分类号 |
C07D307/64;A61K31/341;A61K31/381;A61K31/382;A61K31/4436;A61K31/4535;A61K31/5377;A61P9/00;A61P21/00;A61P25/00;A61P25/28;A61P43/00;C07D233/66;C07D277/32;C07D333/34;C07D333/48;C07D409/12 |
主分类号 |
C07D307/64 |
代理机构 |
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地址 |
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