发明名称 PROCESS FOR THE PREPARATION OF 4- [6-(6-METHANESULFONYL-2-METHYL-PYRIDIN-3-YLAMINO) -5-METHOXY-PYRIMIDIN-4-YLOXY]-PIPERIDINE-1-CARBOXYLIC ACID ISOPROPYL ESTER
摘要 <p>The present invention is directed to a process for the preparation of 4-[6- (6-methanesulfonyl-2-methyl-pyhdin-3-ylamino)-5-methoxy-pyrimidin-4-yloxy]- piperidine-1 -carboxylic acid isopropyl ester, useful as glucose dependent insulinotropic receptor agonist, for the treatment of metabolic-related disorders and complications thereof, such as, diabetes and obesity.</p>
申请公布号 WO2010135506(A1) 申请公布日期 2010.11.25
申请号 WO2010US35538 申请日期 2010.05.20
申请人 JANSSEN PHARMACEUTICA NV;LI, XUN;WELLS, KEN;BRANUM, SHAWN;DAMON, SANDRA 发明人 LI, XUN;WELLS, KEN;BRANUM, SHAWN;DAMON, SANDRA
分类号 C07D401/14;A61K31/506;A61P3/10 主分类号 C07D401/14
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