发明名称 |
PROCESS FOR THE PREPARATION OF 4- [6-(6-METHANESULFONYL-2-METHYL-PYRIDIN-3-YLAMINO) -5-METHOXY-PYRIMIDIN-4-YLOXY]-PIPERIDINE-1-CARBOXYLIC ACID ISOPROPYL ESTER |
摘要 |
<p>The present invention is directed to a process for the preparation of 4-[6- (6-methanesulfonyl-2-methyl-pyhdin-3-ylamino)-5-methoxy-pyrimidin-4-yloxy]- piperidine-1 -carboxylic acid isopropyl ester, useful as glucose dependent insulinotropic receptor agonist, for the treatment of metabolic-related disorders and complications thereof, such as, diabetes and obesity.</p> |
申请公布号 |
WO2010135506(A1) |
申请公布日期 |
2010.11.25 |
申请号 |
WO2010US35538 |
申请日期 |
2010.05.20 |
申请人 |
JANSSEN PHARMACEUTICA NV;LI, XUN;WELLS, KEN;BRANUM, SHAWN;DAMON, SANDRA |
发明人 |
LI, XUN;WELLS, KEN;BRANUM, SHAWN;DAMON, SANDRA |
分类号 |
C07D401/14;A61K31/506;A61P3/10 |
主分类号 |
C07D401/14 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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