发明名称 |
HETEROCYCLIC SULFONAMIDE INHIBITORS OF BETA AMYLOID PRODUCTION |
摘要 |
Compounds of Formula (I), wherein R1, R2, R3, R4, R5, R6, T, W, X, Y and Z are as defined herein are provided, together with pharmaceutically acceptable salt, hydrates and/or prodrugs thereof. Methods of using these compounds for inhibiting beta amyloid production and for treatment of Alzheimer's Disease and Down's syndrome are described. |
申请公布号 |
CA2436526(C) |
申请公布日期 |
2010.10.19 |
申请号 |
CA20012436526 |
申请日期 |
2001.12.11 |
申请人 |
WYETH;ARQULE, INC. |
发明人 |
KREFT, ANTHONY FRANK;COLE, DEREK CECIL;WOLLER, KEVIN ROGER;STOCK, JOSEPH RAYMOND;DIAMANTIDIS, GEORGE;KUBRAK, DENNIS MICHAEL;KUTTERER, KRISTINA MARTHA;MOORE, WILLIAM JAY;CASEBIER, DAVID SCOTT |
分类号 |
C07D333/34;A61K31/341;A61K31/381;A61K31/382;A61K31/4436;A61K31/4535;A61P25/28;A61P43/00;C07D233/66;C07D277/32;C07D307/64;C07D333/48;C07D409/12 |
主分类号 |
C07D333/34 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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