发明名称 INDOL-3-YL-CARBONYL-PIPERIDIN-BENZOIMIDAZOL DERIVATIVES
摘要 The present invention relates to Indol-3-yl-carbonyl-piperidin-benzoimidazol derivatives which act as V1a receptor antagonists and which are represented by Formula I: wherein the residues R1 to R7 are as defined herein. The invention further relates to pharmaceutical compositions containing such compounds, their use in treating dysmenorrhea, hypertension, chronic heart failure, inappropriate secretion of vasopressin, liver cirrhosis, nephritic syndrome, obsessive compulsive disorder, anxiety and depressive disorders, and methods of preparation thereof.
申请公布号 US2010256140(A1) 申请公布日期 2010.10.07
申请号 US20100819243 申请日期 2010.06.21
申请人 BISSANTZ CATERINA;GRUNDSCHOBER CHRISTOPHE;RATNI HASANE;ROGERS-EVANS MARK;SCHNIDER PATRICK 发明人 BISSANTZ CATERINA;GRUNDSCHOBER CHRISTOPHE;RATNI HASANE;ROGERS-EVANS MARK;SCHNIDER PATRICK
分类号 A61K31/454;A61K31/4545;A61K31/5377;A61P1/16;A61P9/00;A61P9/12;A61P13/12;A61P25/00;A61P25/22;A61P25/24;C07D401/14;C07D413/14 主分类号 A61K31/454
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