发明名称 |
INDAZOLE ACRYLIC ACID AMIDE COMPOUND |
摘要 |
A compound of the formula: wherein ring X is benzene or pyridine; R1 is substituted alkyl; R2 is optionally substituted aryl or optionally substituted heterocyclic group; R3 is hydrogen or alkyl; R4 is hydrogen, halogen or alkyl; R5 is hydrogen or alkyl; R6 and R7 are the same or different and each hydrogen or halogen, or a pharmaceutically acceptable salt thereof, which is useful as IKur blocker effective for preventing or treating cardiac arrhythmia such as atrial fibrillation.
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申请公布号 |
US2010256108(A1) |
申请公布日期 |
2010.10.07 |
申请号 |
US20080680497 |
申请日期 |
2008.09.26 |
申请人 |
YAMAGUCHI TETSUO;KAWANISHI HIROYUKI;USHIROGOCHI HIDEKI;TAKAHASHI TATSUYUKI;TAKEBE TOHRU |
发明人 |
YAMAGUCHI TETSUO;KAWANISHI HIROYUKI;USHIROGOCHI HIDEKI;TAKAHASHI TATSUYUKI;TAKEBE TOHRU |
分类号 |
A61K31/437;A61K31/416;A61K31/4439;A61K31/454;A61K31/5377;A61K31/551;A61K31/553;A61P9/06;C07D231/56;C07D401/12;C07D403/12;C07D413/12;C07D471/04 |
主分类号 |
A61K31/437 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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