发明名称 INDAZOLE ACRYLIC ACID AMIDE COMPOUND
摘要 A compound of the formula: wherein ring X is benzene or pyridine; R1 is substituted alkyl; R2 is optionally substituted aryl or optionally substituted heterocyclic group; R3 is hydrogen or alkyl; R4 is hydrogen, halogen or alkyl; R5 is hydrogen or alkyl; R6 and R7 are the same or different and each hydrogen or halogen, or a pharmaceutically acceptable salt thereof, which is useful as IKur blocker effective for preventing or treating cardiac arrhythmia such as atrial fibrillation.
申请公布号 US2010256108(A1) 申请公布日期 2010.10.07
申请号 US20080680497 申请日期 2008.09.26
申请人 YAMAGUCHI TETSUO;KAWANISHI HIROYUKI;USHIROGOCHI HIDEKI;TAKAHASHI TATSUYUKI;TAKEBE TOHRU 发明人 YAMAGUCHI TETSUO;KAWANISHI HIROYUKI;USHIROGOCHI HIDEKI;TAKAHASHI TATSUYUKI;TAKEBE TOHRU
分类号 A61K31/437;A61K31/416;A61K31/4439;A61K31/454;A61K31/5377;A61K31/551;A61K31/553;A61P9/06;C07D231/56;C07D401/12;C07D403/12;C07D413/12;C07D471/04 主分类号 A61K31/437
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