发明名称 |
Dicationic compounds which selectively recognize G-quadruplex DNA |
摘要 |
Dicationic compounds that are highly selective for binding G-quadruplex DNA are described. Several compounds exhibit groove binding toward G-quadruplex DNA and in vitro and in vivo activity versus Trypanosoma brucei rhodesiense. The compounds represent novel drugs for the treatment of cancer, malaria, leishmania, and trypanosomiasis.
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申请公布号 |
US2010249175(A1) |
申请公布日期 |
2010.09.30 |
申请号 |
US20060478453 |
申请日期 |
2006.06.29 |
申请人 |
WILSON W DAVID;BOYKIN DAVID W;WHITE ELIZABETH W;ISMAIL MOHAMED A;KUMAR ARVIND;NANJUNDA RUPESH;TIDWELL RICHARD R |
发明人 |
WILSON W. DAVID;BOYKIN DAVID W.;WHITE ELIZABETH W.;ISMAIL MOHAMED A.;KUMAR ARVIND;NANJUNDA RUPESH;TIDWELL RICHARD R. |
分类号 |
A61K31/437;A61K31/4178;A61P35/04;C07D405/14;C07D471/04;C07H21/04;C12N5/02;C12N5/071;C12P19/34 |
主分类号 |
A61K31/437 |
代理机构 |
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代理人 |
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地址 |
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