发明名称 INHIBITORS OF AKT ACTIVITY
摘要 <p>The instant invention provides for substituted fused naphthyridine derivatives that inhibit Akt activity. In particular, the compounds disclosed selectively inhibit one or two of the Akt isoforms. The invention also provides for compositions comprising such inhibitory compounds and methods of inhibiting Akt activity by administering the compound to a patient in need of treatment of cancer.</p>
申请公布号 WO2010104933(A1) 申请公布日期 2010.09.16
申请号 WO2010US26796 申请日期 2010.03.10
申请人 MERCK SHARP & DOHME CORP.;BANYU PHARMACEUTICAL CO., LTD.;FAN, WEIMING;HAXELL, THOMAS, F. N.;JENKS, MATTHEW, G.;KAWANISHI, NOBUHIKO;LEE, SHULIANG;LIU, HAO;MALASKA, MICHAEL, J.;MOORE, JOSEPH, A., III;OGINO, YOSHIO;ONOZAKI, YU;PANDI, BHARATHI;PEEL, MICHAEL, R.;SAKAMOTO, TOSHIHIRO;SIU, TONY 发明人 FAN, WEIMING;HAXELL, THOMAS, F. N.;JENKS, MATTHEW, G.;KAWANISHI, NOBUHIKO;LEE, SHULIANG;LIU, HAO;MALASKA, MICHAEL, J.;MOORE, JOSEPH, A., III;OGINO, YOSHIO;ONOZAKI, YU;PANDI, BHARATHI;PEEL, MICHAEL, R.;SAKAMOTO, TOSHIHIRO;SIU, TONY
分类号 C07D403/00;C07D413/00 主分类号 C07D403/00
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