发明名称 Nitrogen-containing heteroaryl compounds having inhibitory activity against HIV integrase
摘要 A compound of the formula (I): wherein Z4, Z5 and Z9 each is independently carbon atom or nitrogen atom; Y is hydroxy, mercapto or amino; RA is a group of the formula: (wherein C ring is nitrogen-containing heteroaryl) has an inhibitory activity against integrase.
申请公布号 US7759372(B2) 申请公布日期 2010.07.20
申请号 US20060500387 申请日期 2006.08.08
申请人 SHIONOGI & CO., LTD. 发明人 FUJI MASAHIRO;MIKAMIYAMA HIDENORI;MURAI HITOSHI
分类号 C07D215/48;C07D235/26;A61K31/4184;A61K31/4196;A61K31/422;A61K31/4245;A61K31/427;A61K31/428;A61K31/433;A61K31/4355;A61K31/437;A61K31/47;A61K31/4709;A61K31/498;A61K31/506;A61K31/519;A61K45/00;A61P31/12;A61P31/18;A61P43/00;C07D215/26;C07D215/28;C07D235/06;C07D235/08;C07D235/10;C07D235/18;C07D277/62;C07D277/64;C07D401/04;C07D401/12;C07D403/04;C07D403/06;C07D405/04;C07D405/06;C07D409/06;C07D413/04;C07D413/14;C07D417/04;C07D417/06;C07D417/12;C07D471/04;C07D487/04;C07D491/04;C07D491/048;C07D513/04 主分类号 C07D215/48
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