发明名称 |
BICYCLIC ARYL AND HETEROARYL COMPOUNDS FOR THE TREATMENT OF METABOLIC DISORDERS |
摘要 |
Compounds of formula (I): or pharmaceutically acceptable salts thereof, are opioid receptor modulators, e.g. mu-opioid receptor antagonists, neutral antagonists or inverse agonists, and are useful for the treatment of metabolic disorders including obesity.
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申请公布号 |
US2010173886(A1) |
申请公布日期 |
2010.07.08 |
申请号 |
US20080601100 |
申请日期 |
2008.05.22 |
申请人 |
BLOXHAM JASON;BRADLEY STUART EDWARD;DUPREE TOM BANKSIA;FRY PETER TIMOTHY;HANRAHAN PATRICK ERIC;KRULLE THOMAS MARTIN;PROCTER MARTIN JAMES;SAMBROOK-SMITH COLIN PETER;SCHOFIELD KAREN LESLEY;SMYTH DONALD;STEWART ALAN JOHN |
发明人 |
BLOXHAM JASON;BRADLEY STUART EDWARD;DUPREE TOM BANKSIA;FRY PETER TIMOTHY;HANRAHAN PATRICK ERIC;KRULLE THOMAS MARTIN;PROCTER MARTIN JAMES;SAMBROOK-SMITH COLIN PETER;SCHOFIELD KAREN LESLEY;SMYTH DONALD;STEWART ALAN JOHN |
分类号 |
A61K31/397;A61K31/44;A61K31/47;A61K31/496;A61K31/5377;A61P3/10;A61P9/12;A61P25/24;A61P25/32;A61P25/36;C07D213/84;C07D217/22;C07D403/12;C07D413/12 |
主分类号 |
A61K31/397 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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