发明名称 QUINOLINONE DERIVATIVES AS PARP AND TANK INHIBITORS
摘要 The present invention provides compounds of formula (I), their use as PARP inhibitors as well as pharmaceutical compositions comprising said compounds of formula (I) wherein R1, R2, R3, R4, R5, R6, R7, n, m and X have defined meanings.
申请公布号 US2010168065(A1) 申请公布日期 2010.07.01
申请号 US20080529142 申请日期 2008.03.07
申请人 JANSSEN PHARMACEUTICA NV 发明人 VIALARD JORGE EDUARDO;ANGIBAUD PATRICK RENE;MEVELLEC LAURENCE ANNE;MEYER CHRISTOPHE;FREYNE EDDY JEAN EDGARD;PILATTE ISABELLE NOELLE;ROUX BRUNO;PASQUIER ELISABETH THERESE JEANNE;BOURDREZ XAVIER MARC;ADELINET CHRISTOPHE DENIS;MARCONNET-DECRANE LAURENCE FRANCOISE BERNADETTE;MACRITCHIE JACQUELINE ANNE;DUFFY JAMES EDWARD STEWART;OWENS ANDREW PATE;STORCK PIERRE-HENRI;PONCELET VIRGINIE SOPHIE
分类号 A61K31/675;A61K31/437;A61K31/4704;A61K31/496;A61K31/498;A61K31/502;A61K31/506;A61K31/5377;A61P35/00;C07D215/227;C07D401/12;C07D413/12;C07D471/04;C07F9/38 主分类号 A61K31/675
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