QUINOLINONE DERIVATIVES AS PARP AND TANK INHIBITORS
摘要
The present invention provides compounds of formula (I), their use as PARP inhibitors as well as pharmaceutical compositions comprising said compounds of formula (I) wherein R1, R2, R3, R4, R5, R6, R7, n, m and X have defined meanings.
申请公布号
US2010168065(A1)
申请公布日期
2010.07.01
申请号
US20080529142
申请日期
2008.03.07
申请人
JANSSEN PHARMACEUTICA NV
发明人
VIALARD JORGE EDUARDO;ANGIBAUD PATRICK RENE;MEVELLEC LAURENCE ANNE;MEYER CHRISTOPHE;FREYNE EDDY JEAN EDGARD;PILATTE ISABELLE NOELLE;ROUX BRUNO;PASQUIER ELISABETH THERESE JEANNE;BOURDREZ XAVIER MARC;ADELINET CHRISTOPHE DENIS;MARCONNET-DECRANE LAURENCE FRANCOISE BERNADETTE;MACRITCHIE JACQUELINE ANNE;DUFFY JAMES EDWARD STEWART;OWENS ANDREW PATE;STORCK PIERRE-HENRI;PONCELET VIRGINIE SOPHIE