发明名称 1, 3, 5 -TRIAZ INE DERIVATIVES USEFUL IN THE TREATMENT OF CHRONIC PAIN DISORDERS
摘要 The present invention provides compounds that are inhibitors of voltage-gated sodium channel (Nav), in particular Nav 1.7 and are therefore useful for the treatment of diseases 5 treatable by inhibition of these channels, in particular, chronic pain disorders. Also provided are pharmaceutical compositions containing such compounds and processes for preparing such compounds.
申请公布号 WO2010022055(A3) 申请公布日期 2010.06.17
申请号 WO2009US54169 申请日期 2009.08.18
申请人 AMGEN INC.;BUCHANAN, JOHN L.;BREGMAN, HOWARD;CHAKKA, NAGASREE;DIMAURO, ERIN F.;DU, BINGFAN;NGUYEN, HANH NHO;ZHENG, XIAO MEI 发明人 BUCHANAN, JOHN L.;BREGMAN, HOWARD;CHAKKA, NAGASREE;DIMAURO, ERIN F.;DU, BINGFAN;NGUYEN, HANH NHO;ZHENG, XIAO MEI
分类号 C07D401/04;A61K31/53;A61P25/04;C07D401/12;C07D401/14;C07D471/04 主分类号 C07D401/04
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