发明名称 TECHNETIUM-AND RHENIUM-BIS(HETEROARYL)COMPLEXES AND METHODS OF USE THEREOF
摘要 Complexes of heterocyclic radionuclides are prepared based upon ligands having substituted pyridyl and imidazolyl groups. The ligands are bifunctional, having amino acid residues that may act as a linker to a bioactive molecule, and a tridentate chelator that may complex the radionuclide. The bioactive molecule may be a peptide or somatostatin.
申请公布号 WO2010065899(A2) 申请公布日期 2010.06.10
申请号 WO2009US66832 申请日期 2009.12.04
申请人 MOLECULAR INSIGHT PHARMACEUTICALS, INC.;BABICH, JOHN, W.;ZIMMERMAN, CRAIG;JOYAL, JOHN;MARESCA, KEVIN, P.;MARQUIS, JOHN;LU, GENLIANG;WANG, JIAN-CHENG;HILLIER, SHAWN 发明人 BABICH, JOHN, W.;ZIMMERMAN, CRAIG;JOYAL, JOHN;MARESCA, KEVIN, P.;MARQUIS, JOHN;LU, GENLIANG;WANG, JIAN-CHENG;HILLIER, SHAWN
分类号 C07D213/38;A61K51/04;A61K51/08;C07F13/00 主分类号 C07D213/38
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