发明名称 PROCESS FOR THE PREPARATION OF SUBSTANTIALLY OPTICALLY PURE REPAGLINIDE AND PRECURSORS THEREOF
摘要 <p>The invention relates to a process for preparing substantially optically pure repaglinide and pharmaceutically acceptable salts, solvates and esters thereof. The invention further relates to a process for preparing precursors of repaglinide and in particular for preparing ( S ) ( f ) - 1 - ( 2 -piperidino-phenyl ) -3 - methyl - I -butylamine.</p>
申请公布号 WO2010046360(A1) 申请公布日期 2010.04.29
申请号 WO2009EP63734 申请日期 2009.10.20
申请人 KRKA, TOVARNA ZDRAVIL, D.D., NOVO MESTO;VEVERKA, MIROSLAV;VEVERKOVA, EVA;KLVANOVA, JANA;BOMBEK, SERGEJA;MERSLAVIC, MARJO;SMODIS, JANEZ 发明人 VEVERKA, MIROSLAV;VEVERKOVA, EVA;KLVANOVA, JANA;BOMBEK, SERGEJA;MERSLAVIC, MARJO;SMODIS, JANEZ
分类号 A61K31/4453;A61P5/50;C07D295/135 主分类号 A61K31/4453
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