HETEROCYCLYL AND CYCLOALKYL SUBSTITUTED THIENO [2,3-D] PYRIMIDINE AND THEIR USE AS ADENOSINE A2A RECEPTOR ANTAGONISTS
摘要
<p>This invention relates to a novel thieno[2,3-d]pyrimidine, Z, and its therapeutic and prophylactic uses, wherein X, R1 and R2 are defined in the specification. Disorders treatedand/or prevented include Parkinson's Disease.Formula (I).</p>
申请公布号
WO2010045016(A1)
申请公布日期
2010.04.22
申请号
WO2009US58738
申请日期
2009.09.29
申请人
JANSSEN PHARMACEUTICA NV;BARBAY, J. KENT;LEONARD, KRISTI;CHAKRAVARTY, DEVRAJ;SHOOK, BRIAN, CHRISTOPHER;WANG, AIHUA
发明人
BARBAY, J. KENT;LEONARD, KRISTI;CHAKRAVARTY, DEVRAJ;SHOOK, BRIAN, CHRISTOPHER;WANG, AIHUA