发明名称 NOVEL CRYSTALLINE COMPOUND USEFUL AS GLK ACTIVATOR
摘要 A novel crystalline form of 3-{[5-(azetidin-1-ylcarbonyl)pyrazin-2-yl]oxy}-5-[(1-methylethyl)oxy]-N-1H-pyrazol-3-ylbenzamide is described in the specification. This compound is a glucokinase (GLK or GK) activator and useful as a pharmaceutical agent in the treatment or prevention of a disease or medical condition mediated through GLK, leading to a decreased glucose threshold for insulin secretion. Processes for the manufacture of the crystalline form, pharmaceutical compositions comprising the crystalline form and the use of the crystalline form in medical treatment are also described.
申请公布号 US2010094009(A1) 申请公布日期 2010.04.15
申请号 US20070520223 申请日期 2007.12.20
申请人 MCCABE JAMES;TOMKINSON GARY PETER 发明人 MCCABE JAMES;TOMKINSON GARY PETER
分类号 C07D401/14 主分类号 C07D401/14
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