发明名称 |
ATP-BINDING CASETTE TRANSPORTER MODULATORS |
摘要 |
FIELD: chemistry. ^ SUBSTANCE: novel compound is N-(5-hydroxy-2,4-di-tert-butylphenyl)-4-oxo-1H-quinoline-3-carboxamide or its pharmaceutically acceptable salts. The invention also relates to a pharmaceutical composition. ^ EFFECT: obtaining a novel biologically active compound with CFTR activity modulation properties. ^ 2 cl, 485 ex, 3 tbl |
申请公布号 |
RU2382779(C2) |
申请公布日期 |
2010.02.27 |
申请号 |
RU20070102578 |
申请日期 |
2005.06.24 |
申请人 |
VERTEKS FARMAS'JUTIKALZ INKORPOREJTED |
发明人 |
ADIDA RUA SARA S.;KHEJZLVUD ANNA R.;GROTENKHEJS PETER D. J.;VAN GUR FREDERIK F.;SINGKH ASHVANI K.;CHZHOU TSZINLAN';MAKKARTNI DZHEJSON |
分类号 |
A61K31/47;A61K31/4709;A61P25/00;A61P31/00;C07D209/12;C07D209/14;C07D209/18;C07D215/56;C07D401/12;C07D405/12;C07D409/12;C07D413/12;C07D417/12 |
主分类号 |
A61K31/47 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|