发明名称 |
FOSAPREPITANT DIMEGLUMINE INTERMEDIATE, NEUTRAL FOSAPREPITANT, AND AMORPHOUS FOSAPREPITANT DIMEGLUMINE AND PROCESSES FOR THEIR PREPARATIONS |
摘要 |
<p>The present invention generally relates to a process for the preparation of fosaprepitant dimeglumine intermediate and its use in the preparation of fosaprepitant dimeglumine; to a neutral form of fosaprepitant in a solid state and processes for the preparation thereof; and to a stable amorphous fosaprepitant dimeglumine, having a stability at temperatures of about 2°C to about 8°C and at a relative humidity below at least 60%; and a process for the preparation thereof.</p> |
申请公布号 |
CA2730681(A1) |
申请公布日期 |
2010.02.18 |
申请号 |
CA20092730681 |
申请日期 |
2009.07.17 |
申请人 |
GLENMARK GENERICS LIMITED |
发明人 |
GANESHBHATT, NAVIN;RASIKLALTRIVEDI, NIKHIL;KHEDEKAR, MAHESH;SINHA, SUKUMAR;AHMED KHAN, MUBEEN;YADAV, RAMJILAL |
分类号 |
C07F9/40 |
主分类号 |
C07F9/40 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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