发明名称 PRODRUGS OF FUSED HETEROCYCLIC INHIBITORS OF D-AMINO ACID OXIDASE
摘要 <p>The invention relates to prodrugs of fused heterocyclic inhibitors of D-amino oxidase (DAAO) and methods of treating diseases and conditions, wherein modulation of D- amino acid oxidase activity, D-serine levels, D-serine oxidative products and NMDA receptor activity in the nervous system of a mammalian subject is effective.</p>
申请公布号 WO2010017418(A1) 申请公布日期 2010.02.11
申请号 WO2009US53049 申请日期 2009.08.06
申请人 SEPRACOR INC.;HEFFERNAN, MICHELE, L.R.;DENNIS, RICHARD;DORSEY, JAMES, M.;FOGLESONG, ROBERT, J.;JONES, MICHAEL, L.;OGBU, CYPRIAN, O.;SOUKRI, MUSTAPHA;SPEAR, KERRY, L.;WILKINSON, H., SCOTT;ORSINI, MICHAEL ANTHONY 发明人 HEFFERNAN, MICHELE, L.R.;DENNIS, RICHARD;DORSEY, JAMES, M.;FOGLESONG, ROBERT, J.;JONES, MICHAEL, L.;OGBU, CYPRIAN, O.;SOUKRI, MUSTAPHA;SPEAR, KERRY, L.;WILKINSON, H., SCOTT;ORSINI, MICHAEL ANTHONY
分类号 A61K31/407;C07D491/04;A61P25/00 主分类号 A61K31/407
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