发明名称 ACID ADDITION SALTS OF IMATINIB AND FORMULATIONS COMPRISING THE SAME
摘要 Acid addition salts of 4-[(4-Methyl-1-piperazinyl)methyl]-N-[4-methyl-3-[[4-(3-pyridinyl)-2-pyrimidinyl]amino]phenyl]-benzamide selected from the group consisting of an orotate salt, an oxalate salt, a nicotinate salt, a camphor sulfonate salt, a para-toluene sulfonate salt, a laurate salt, an aspartate salt, a caprate salt, an oleate salt and a phenyl acetate salt is disclosed. The invention further provides a method for producing said acid addition salts and formulations, preferably solid formulations comprising at least one of said salts within the composition.
申请公布号 WO2009065910(A3) 申请公布日期 2009.12.30
申请号 WO2008EP65943 申请日期 2008.11.20
申请人 ZENTIVA KIMYASAL URUNLER SANAYI VE TICARET A.S.;ADIYAMAN, MUSTAFA;DURMUS, SEMIH;SAHPAZ CERIT, FILIZ 发明人 ADIYAMAN, MUSTAFA;DURMUS, SEMIH;SAHPAZ CERIT, FILIZ
分类号 A61K31/505;A61P35/00 主分类号 A61K31/505
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