发明名称 |
ACID ADDITION SALTS OF IMATINIB AND FORMULATIONS COMPRISING THE SAME |
摘要 |
Acid addition salts of 4-[(4-Methyl-1-piperazinyl)methyl]-N-[4-methyl-3-[[4-(3-pyridinyl)-2-pyrimidinyl]amino]phenyl]-benzamide selected from the group consisting of an orotate salt, an oxalate salt, a nicotinate salt, a camphor sulfonate salt, a para-toluene sulfonate salt, a laurate salt, an aspartate salt, a caprate salt, an oleate salt and a phenyl acetate salt is disclosed. The invention further provides a method for producing said acid addition salts and formulations, preferably solid formulations comprising at least one of said salts within the composition. |
申请公布号 |
WO2009065910(A3) |
申请公布日期 |
2009.12.30 |
申请号 |
WO2008EP65943 |
申请日期 |
2008.11.20 |
申请人 |
ZENTIVA KIMYASAL URUNLER SANAYI VE TICARET A.S.;ADIYAMAN, MUSTAFA;DURMUS, SEMIH;SAHPAZ CERIT, FILIZ |
发明人 |
ADIYAMAN, MUSTAFA;DURMUS, SEMIH;SAHPAZ CERIT, FILIZ |
分类号 |
A61K31/505;A61P35/00 |
主分类号 |
A61K31/505 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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