发明名称 |
PROCESS FOR THE SYNTHESIS OF DERIVATIVES OF 3-AMINO-TETRAHYDROFURAN-3-CARBOXYLIC ACID AND USE THEREOF AS MEDICAMENTS |
摘要 |
The present invention relates to a process for the manufacturing of substituted 3-amino-tetrahydrofuran-3-carboxylic acid amides of general formula (I) and their precursors in high optical purity to the precursors of the synthesis of substituted S-Amino-tetrahydrofuran-S-carboxylic acid amides of general formula (I) in high optical purity, and to the tautomers, enantiomers, diastereomers, mixtures and salts of substituted 3-amino-tetrahydrofuran-3-carboxylic acid amides of general formula (I) in high optical purity, particularly the physiologically acceptable salts thereof with inorganic or organic acids or bases, which have valuable properties.
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申请公布号 |
KR20090097208(A) |
申请公布日期 |
2009.09.15 |
申请号 |
KR20097016217 |
申请日期 |
2007.12.21 |
申请人 |
BOEHRINGER INGELHEIM INTERNATIONAL GMBH |
发明人 |
HAN ZHENGXU;GERLACH KAI;KRISHNAMURTHY DHILEEPKUMAR;MATTHES BURKHARD;NAR HERBERT;PFAU ROLAND;PRIEPKE HENNING;SCHULER METZ ANNETTE;SENANAYAKE CHRIS H.;SIEGER PETER;TANG WENJUN;WIENEN WOLFGANG;XU YIBO;YEE NATHAN K. |
分类号 |
C07D413/14;C07D307/24;C07D409/14 |
主分类号 |
C07D413/14 |
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