摘要 |
THE PRESENT INVENTION RELATES TO A PROCESS FOR PREPARING 5-CHLORO-N-({(5S)-2-OXO-3-[4-(3-OXO-4-MORPHOLINYL)PHENYL]-1,3-OXAZOLIDIN-5- YL} METHYL)-2-THIOPHENECARBOXAMIDE STARTING FROM 2-[(2S)-2-OXIRANYLMETHYL]-IH-ISOINDOLE-1,3(2H)-DIONE, 4-( 4-AMINOPHENYL)- 3-MORPHOLINONE AND 5-CHLOROTHIOPHENE-2-CARBONYL CHLORIDE.
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