发明名称 RENIN INHIBITORS
摘要 <p>Disclosed are compounds having the formula (I): wherein the R1, R2, R3, X, Y, A, L, and G are defined herein. These compounds bind to aspartic proteases to inhibit their activity and are useful in the treatment or amelioration of diseases associated with aspartic protease activity. Also disclosed are methods of use of the compounds of Formula I for ameliorating or treating aspartic protease related disorders in a subject in need thereof.</p>
申请公布号 WO2009096996(A1) 申请公布日期 2009.08.06
申请号 WO2008US67650 申请日期 2008.06.20
申请人 SMITHKLINE BEECHAM CORPORATION;VITAE PHARMACEUTICALS, INC.;BALDWIN, JOHN J.;CACATIAN, SALVACION;CLAREMON, DAVID;DILLARD, LAWRENCE, W.;FLAHERTY, PATRICK, T.;GHAVIMI-ALAGHA, BAHMAN;ISHCHENKO, ALEXEY, V.;GHIRLANDA, DAMIANO;KALLANDER, LARA, S.;LAWHORN, BRIAN;LU, QING;MCGEEHAN, GERARD;KNAPP-REED, BETH, A.;SEMUS, SIMON;SIMPSON, ROBERT, D.;SINGH, SURESH, B.;TERRELL, LAMONT, R.;TICE, COLIN;TRAN, TRITIN;XU, ZHENRONG;YUAN, JING;ZHAO, WEI;ZHAO, YONGDONG Y. 发明人 BALDWIN, JOHN J.;CACATIAN, SALVACION;CLAREMON, DAVID;DILLARD, LAWRENCE, W.;FLAHERTY, PATRICK, T.;GHAVIMI-ALAGHA, BAHMAN;ISHCHENKO, ALEXEY, V.;GHIRLANDA, DAMIANO;KALLANDER, LARA, S.;LAWHORN, BRIAN;LU, QING;MCGEEHAN, GERARD;KNAPP-REED, BETH, A.;SEMUS, SIMON;SIMPSON, ROBERT, D.;SINGH, SURESH, B.;TERRELL, LAMONT, R.;TICE, COLIN;TRAN, TRITIN;XU, ZHENRONG;YUAN, JING;ZHAO, WEI;ZHAO, YONGDONG Y.
分类号 C09K11/06 主分类号 C09K11/06
代理机构 代理人
主权项
地址