发明名称 |
SOLID FORMS OF 3-(6-(1-(2,2-DIFLUOROBENZO[D][1,3] DIOXOL-5-YL) CYCLOPROPANECARBOXAMIDO)-3-METHYLPYRIDIN-2-YL) BENZOIC ACID |
摘要 |
The present invention relates to a substantially crystalline and free solid state form of 3-(6-(l-(2,2-difluorobenzo[d][l,3]dioxol-5-yl) cyclopropanecarboxamido)-3- methylPyridin-2-yl)benzoic acid (Form I) of following formula: (I), pharmaceutical compositions thereof, and methods of treatment therewith. |
申请公布号 |
WO2009073757(A1) |
申请公布日期 |
2009.06.11 |
申请号 |
WO2008US85456 |
申请日期 |
2008.12.04 |
申请人 |
VERTEX PHARMACEUTICALS INCORPORATED;KESHAVARZ-SHOKRI, ALI;ZHANG, BEILI;KRAWIEC, MARIUSZ |
发明人 |
KESHAVARZ-SHOKRI, ALI;ZHANG, BEILI;KRAWIEC, MARIUSZ |
分类号 |
C07D405/12;A61K31/443;A61P11/00 |
主分类号 |
C07D405/12 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|