METHOD FOR THE PRODUCTION OF 17 ALPHA-ACETOXY-6-METHYLENEPREGN-4-ENE-3,20-DIONE, MEDROXYPROGESTERONE ACETATE, AND MEGESTROL ACETATE
摘要
The invention relates to a method for producing 17a-acetoxy-6-methylenepregn-4-ene-3,20-dione (4) as an intermediate preparation as well as methods for producing medroxyprogesterone acetate (1) (17a-acetoxy-6a-methylpregn-4-ene-3,20-dione) and megestrol acetate (2) (17a-acetoxy-6-methylpregna-4,6-diene-3,20-dione) via said intermediate preparation (4).
申请公布号
WO2008148473(A3)
申请公布日期
2009.06.04
申请号
WO2008EP04156
申请日期
2008.05.24
申请人
BAYER SCHERING PHARMA AG;ANNEN, KLAUS;LINZ, THOMAS;NEFF, KARL-HEINZ;BOHLMANN, ROLF;LAURENT, HENRY
发明人
ANNEN, KLAUS;LINZ, THOMAS;NEFF, KARL-HEINZ;BOHLMANN, ROLF;LAURENT, HENRY