| 摘要 |
Disclosed is 1-(2-(4-((2,3-dihydro(1,4)dioxino(2,3-c)pyridin-7-ylmethyl)amino)piperidin-1-yl)ethyl)-7-fluoro-1,5-naphthyridin-2(1H)-one monohydrate, which has a strong antibacterial activity. The compound is highly safe and useful as an original drug for pharmaceutical preparations. Also disclosed is a method which is useful for producing 1-(2-(4-((2,3-dihydro(1,4)dioxino(2,3-c)pyridin-7-ylmethyl)amino)piperidin-1-yl)ethyl)-7-fluoro-1,5-naphthyridin-2(1H)-one monohydrate.
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| 申请人 |
TOYAMA CHEMICAL CO., LTD.;TAISHO PHARMACEUTICAL CO., LTD.;KIYOTO, TARO;TAKEBAYASHI, MASAHIRO;BABA, YASUTAKA;SYOJI, MUNEO;NOGUCHI, TOSHIYA;USHIYAMA, FUMIHITO;URABE, HIROKI;HORIKIRI, HIROMASA |
发明人 |
KIYOTO, TARO;TAKEBAYASHI, MASAHIRO;BABA, YASUTAKA;SYOJI, MUNEO;NOGUCHI, TOSHIYA;USHIYAMA, FUMIHITO;URABE, HIROKI;HORIKIRI, HIROMASA |
