发明名称 QUINAZOLINONE DERIVATIVES, THE PREPARATION METHODS AND USES THEREOF
摘要 <p>The quinzolinone derivatives, the preparation methods and uses thereof. The quinzolinone compounds having the structure of general formula (I), or their pharmaceutical acceptable salts. Most of these compounds have strong activities of inhibiting PDE5, and have highly selectivity of PDE 6 which is distributed on the retina. So the present compounds are expected to exhibit good safety and effectiveness and have broad uses in clinic.</p>
申请公布号 WO2009062402(A1) 申请公布日期 2009.05.22
申请号 WO2008CN01859 申请日期 2008.11.07
申请人 TOPHARMAN SHANGHAI CO., LTD.;SHANGHAI INSTITUTE OF MATERIA MEDICA, CHINESE ACADEMY OF SCIENCES;SHEN, JINGSHAN;ZHENG, JIN;LAI, QINGLIN;WANG, ZHEN;ZHANG, JINFENG;TIAN, GUANGHUI;DUAN, HONGLIANG 发明人 SHEN, JINGSHAN;ZHENG, JIN;LAI, QINGLIN;WANG, ZHEN;ZHANG, JINFENG;TIAN, GUANGHUI;DUAN, HONGLIANG
分类号 A61K31/505;C07D239/91;A61K31/517;A61P9/12;A61P11/08;A61P13/08;A61P13/10;A61P15/00;A61P15/14;A61P27/06;A61P29/00;C07C237/42 主分类号 A61K31/505
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