发明名称 BENZOTHIAZOLE COMPOUNDS
摘要 The present invention relates to benzothiazole compounds that mimic the activity of BH3 only proteins and are capable of binding to and neutralizing pro survival Bcl 2 proteins. The invention also relates to the use of such compounds in the regulation of cell death or cell survival and the treatment and/or prophylaxis of diseases or conditions associated with the deregulation of cell death or cell survival.
申请公布号 WO2009039553(A1) 申请公布日期 2009.04.02
申请号 WO2007AU01442 申请日期 2007.09.27
申请人 THE WALTER AND ELIZA HALL INSTITUTE OF MEDICAL RESEARCH;WATSON, KEITH GEOFFREY;LESSENE, GUILLAUME LAURENT;BAELL, JONATHAN BAYLDON;HUANG, DAVID CHING SIANG;STREET, IAN PHILIP;ADAMS, JERRY MCKEE;COLMAN, PETER MALCOLM;SLEEBS, BRAD EDMUND;SMITH, BRIAN JOHN;CZABOTAR, PETER EDWARD 发明人 WATSON, KEITH GEOFFREY;LESSENE, GUILLAUME LAURENT;BAELL, JONATHAN BAYLDON;HUANG, DAVID CHING SIANG;STREET, IAN PHILIP;ADAMS, JERRY MCKEE;COLMAN, PETER MALCOLM;SLEEBS, BRAD EDMUND;SMITH, BRIAN JOHN;CZABOTAR, PETER EDWARD
分类号 C07D277/82;A61K31/428;A61P19/02;A61P29/00;A61P35/02;A61P37/06;C07D417/12;C07D417/14 主分类号 C07D277/82
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