发明名称 N-(4-(imidazo[1,2A]pyridin-YL)phenethyl)benzamide inhibitors of the mitotic kinesin CENP-E for treating certain cellular proliferation diseases
摘要 Provided herein are certain substituted N-phenethylbenzamide of formula V: that may be useful for treating certain cellular proliferation diseases and disorders by modulating the activity of CENP-E.
申请公布号 US7504413(B2) 申请公布日期 2009.03.17
申请号 US20050271147 申请日期 2005.11.09
申请人 CYTOKINETICS, INC.;SMITHKLINE BEECHAM CORPORATION 发明人 QIAN XIANGPING;BERGNES GUSTAVE;DHANAK DASHYANT;KNIGHT STEVEN D.;ADAMS NICHOLAS D.;PARRISH CYNTHIA A.
分类号 C07D471/02;A61K31/4184;A61K31/4196;A61K31/421;A61K31/424;A61K31/4439;A61K31/4745;A61K31/55;C07C235/48;C07C235/50;C07C235/52;C07C237/22;C07C255/57;C07C257/18;C07C259/18;C07C271/20;C07C271/28;C07C275/40;C07C281/06;C07C311/37;C07D207/26;C07D207/273;C07D211/76;C07D213/30;C07D231/12;C07D235/18;C07D235/26;C07D261/08;C07D263/10;C07D271/06;C07D277/56;C07D285/02;C07D295/155;C07D333/38;C07D403/10;C07D403/12;C07D471/04;C07D487/02;C07D491/02;C07F9/6506;C07F9/6561 主分类号 C07D471/02
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