发明名称 NOVEL ANTI-INFLAMMATORY ANDROSTANE DERIVATIVES.
摘要 THERE ARE PROVIDED COMPOUND OF FORMULA (I) WHEREIN R1 REPRESENTS C1-6 ALKYL OR C1-6 HALOALKYL; R2 REPRESENTS C3-8 CYCLOALKYL OR C3-8 CYCLOALKENYL EITHER OF WHICH MAY OPTIONALLY BE SUBSTITUTED BY ONE OR MORE GROUPS SELECTED FROM OXO, METHYL, METHYLENE AND HALOGEN; R3 REPRESENTS HYDROGEN, METHYL (WHICH MAY BE IN EITHER THE a OR b CONFIGURATION) OR METHYLENE; R4 AND R5 ARE THE SAME OR DIFFERENT AND EACH REPRESENTS HYDROGEN OR HALOGEN; AND ------ REPRESENTS A SINGLE OR A DOUBLE BOND; AND SOLVATES THEREOF, PROCESSES FOR PREPARING THEM AND THEIR USE IN THERAPY.
申请公布号 MY137522(A) 申请公布日期 2009.02.27
申请号 MYPI20021593 申请日期 2002.04.30
申请人 GLAXO GROUP LIMITED 发明人 KEITH BIGGADIKE;PAUL JONES;JEREMY JOHN PAYNE
分类号 A61K9/12;A61K9/72;A61K31/18;A61K31/569;A61K45/00;A61P1/04;A61P5/44;A61P11/00;A61P11/02;A61P11/06;A61P17/00;A61P17/04;A61P17/06;A61P19/02;A61P27/14;A61P27/16;A61P29/00;A61P37/08;A61P43/00;C07J31/00 主分类号 A61K9/12
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