发明名称 INTRAVENOUS AND ORAL DOSING OF A DIRECT-ACTING AND REVERSIBLE P2Y12 INHIBITOR
摘要 The invention provides methods and compositions for rapid and reversible inhibition of platelet aggregation in human subjects in need thereof by administering compounds of the formula: (I) alone or in combination with a second agent which can be aspirin or a thrombolytic agent.
申请公布号 WO2008137753(A3) 申请公布日期 2009.02.12
申请号 WO2008US62518 申请日期 2008.05.02
申请人 PORTOLA PHARMACEUTICALS, INC.;SCARBOROUGH, CARROLL, ANNA, CREW;GRETLER, DANIEL, D.;CONLEY, PAMELA, B.;ANDRE, PATRICK;HUTCHALEELAHA, ATHIWAT;PHILLIPS, DAVID, R.;PANDEY, ANJALI;WOLIN, HUANG 发明人 GRETLER, DANIEL, D.;CONLEY, PAMELA, B.;ANDRE, PATRICK;HUTCHALEELAHA, ATHIWAT;PHILLIPS, DAVID, R.;PANDEY, ANJALI;WOLIN, HUANG;SCARBOROUGH, ROBERT, M.
分类号 A61K31/216;A61K31/517;A61P7/02 主分类号 A61K31/216
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