发明名称 PROCESS FOR THE SYNTHESIS OF DERIVATIVES OF 3-AMINO-TETRAHYDROFURAN-3-CARBOXYLIC ACID AND USE THEREOF AS MEDICAMENTS
摘要 The present invention relates to a process for the manufacturing of subst ituted 3- amino-tetrahydrofuran-3-carboxylic acid amides of general formula (I) and their precursors in high optical purity to the precursors of the syn thesis of substituted S-Amino-tetrahydrofuran-S-carboxylic acid amides of ge neral formula (I) in high optical purity, and to the tautomers, enantiomers, diastereomers, mixtures and salts of substituted 3-amino- tetrahydrofuran-3 -carboxylic acid amides of general formula (I) in high optical purity, parti cularly the physiologically acceptable salts thereof with inorganic or organ ic acids or bases, which have valuable properties.
申请公布号 CA2674168(A1) 申请公布日期 2008.07.10
申请号 CA20072674168 申请日期 2007.12.21
申请人 BOEHRINGER INGELHEIM INTERNATIONAL GMBH 发明人 PFAU, ROLAND;PRIEPKE, HENNING;SCHULER-METZ, ANNETTE;KRISHNAMURTHY, DHILEEPKUMAR;SIEGER, PETER;SENANAYAKE, CHRIS H.;HAN, ZHENGXU;GERLACH, KAI;WIENEN, WOLFGANG;TANG, WENJUN;YEE, NATHAN K.;XU, YIBO;MATTHES, BURKHARD;NAR, HERBERT
分类号 C07D307/24;C07D409/14;C07D413/14 主分类号 C07D307/24
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