发明名称 MACROCYCLIC COMPOUND USEFUL AS PHARMACEUTICAL
摘要 <p><P>PROBLEM TO BE SOLVED: To provide a new analogue of F152. <P>SOLUTION: The invention provides compounds having formula (I), and methods for the synthesis of the compounds and methods for treatment of various disorders (including inflammatory disorders, autoimmune disorders, malignancy and disorders involving increased vascular system formation), the compounds can be used in prevention of restenosis of blood vessel exposed to trauma (for example, angioplasty and stenting). <P>COPYRIGHT: (C)2009,JPO&INPIT</p>
申请公布号 JP2008297317(A) 申请公布日期 2008.12.11
申请号 JP20080194192 申请日期 2008.07.28
申请人 EISAI R & D MANAGEMENT CO LTD 发明人 BOIVIN ROCH;CHIBA KENICHI;DU HONG;EGUCHI YOSHIHITO;FUJITA MASANORI;GOTO MASAKI;HARMANGE JEAN CHRISTOPHE;INOUE ATSUSHI;JIANG YIMIN;KAWADA MEGUMI;KAWAI TAKATOSHI;KAWAKAMI YOSHIYUKI;KIMURA AKIFUMI;KOTAKE MAKOTO;KUBOI YOSHIKAZU;LEMELIN CHARLES-ANDRE;LI XIANG-YI;MATSUSHIMA TOMOHIRO;MIZUI YOSHIHARU;SAKURAI HIDEKI;SHEN YONGCHUN;SPYVEE MARK;TANAKA ISAO;WANG JOHN (YUAN);YAMAMOTO SOJI;YONEDA NAOKI;CHOW JESSE;GUSOVSKY FABIAN;MURAMOTO KENZO;SHIROTA HIROSHI
分类号 C07D313/00;C07D491/044;A61K31/335;A61K31/36;A61K31/365;A61K31/395;A61K31/4178;A61K31/4188;A61K31/5377;A61P1/00;A61P1/04;A61P1/16;A61P3/10;A61P7/04;A61P9/00;A61P9/10;A61P11/00;A61P11/02;A61P11/06;A61P11/08;A61P13/02;A61P17/00;A61P17/04;A61P17/06;A61P17/16;A61P19/02;A61P19/04;A61P19/10;A61P21/04;A61P25/00;A61P25/02;A61P25/08;A61P25/28;A61P27/02;A61P29/00;A61P31/04;A61P31/18;A61P33/06;A61P35/00;A61P35/02;A61P37/02;A61P37/06;A61P37/08;A61P43/00;C07D267/00;C07D401/12;C07D405/12;C07D491/04;C07D491/08;C07D493/04;C07D521/00 主分类号 C07D313/00
代理机构 代理人
主权项
地址