发明名称 MUTILIN DERIVATIVES AND THEIR USE AS PHARMACEUTICAL
摘要 14-0-[(((C1.6)Alkoxy-(C1.6)alkyl)-phenylsulfanyl)-acetyl]-mutilins, 14-O-[(((C1-6)Mono-or dialkylamino-(C1.6)alkyl)-phenylsulfanyl)-acetyl]-mutilins, 14-O-[((Hydroxy-(C1-6)-alkyl)-phenylsulfanyl)-acetyl]-mutilins, 14-O-[((Formyl-(C0.5)-alkyl)-phenylsulfanyl)-acetyl]-mutilins, 14-O-[((Guanidino-imino-(C1-6)alkyl)-phenylsulfanyl)-acetyl]-mutilins, 14-O-[((Ureido-imino-(C1-6)alky)-phenylsulfany]-acety]-mutilins, 14-O-[((Thioureido-imino-(C1-6)alkyl)-phenylsulfanyl)-acetyl]-mutilins, 14-O-[((lsothioureido-imino-(C1-6)alkyl)-phenylsulfanyl)-acetyl]-mutilins and their use as pharmaceuticals. ® KIPO & WIPO 2009
申请公布号 KR20080104273(A) 申请公布日期 2008.12.02
申请号 KR20087019893 申请日期 2007.01.11
申请人 NABRIVA THERAPEUTICS AG 发明人 THIRRING KLAUS;ASCHER GERD;PAUKNER SUSANNE;HEILMAYER WERNER;NOVAK RODGER
分类号 C07C323/52;A61K31/22;C07D295/20;C07D295/215 主分类号 C07C323/52
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