发明名称 PREPARATION OF RIVASTIGMINE AND ITS SALTS
摘要 There are provided processes for making rivastigmine. In one embodiment, the process includes reacting S-(-)-[1-(3-hydroxyphenyl)ethyl]dimethylamine with N-ethyl-N-methyl carbamoyl chloride in the presence of an organic base to obtain a free base of rivastigmine.
申请公布号 US2008255383(A1) 申请公布日期 2008.10.16
申请号 US20080100591 申请日期 2008.04.10
申请人 MANDAVA VENKATA NAGA BRAHMESWARA RAO;VAJRALA VENKATA REDDY;VARANASI GANESH;ADLA VIJAY KUMAR;JAMBULA MUKUND REDDY;KANUMATHI REDDY VIJAYPAL REDDY 发明人 MANDAVA VENKATA NAGA BRAHMESWARA RAO;VAJRALA VENKATA REDDY;VARANASI GANESH;ADLA VIJAY KUMAR;JAMBULA MUKUND REDDY;KANUMATHI REDDY VIJAYPAL REDDY
分类号 C07C269/00 主分类号 C07C269/00
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