发明名称 |
PREPARATION OF RIVASTIGMINE AND ITS SALTS |
摘要 |
There are provided processes for making rivastigmine. In one embodiment, the process includes reacting S-(-)-[1-(3-hydroxyphenyl)ethyl]dimethylamine with N-ethyl-N-methyl carbamoyl chloride in the presence of an organic base to obtain a free base of rivastigmine.
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申请公布号 |
US2008255383(A1) |
申请公布日期 |
2008.10.16 |
申请号 |
US20080100591 |
申请日期 |
2008.04.10 |
申请人 |
MANDAVA VENKATA NAGA BRAHMESWARA RAO;VAJRALA VENKATA REDDY;VARANASI GANESH;ADLA VIJAY KUMAR;JAMBULA MUKUND REDDY;KANUMATHI REDDY VIJAYPAL REDDY |
发明人 |
MANDAVA VENKATA NAGA BRAHMESWARA RAO;VAJRALA VENKATA REDDY;VARANASI GANESH;ADLA VIJAY KUMAR;JAMBULA MUKUND REDDY;KANUMATHI REDDY VIJAYPAL REDDY |
分类号 |
C07C269/00 |
主分类号 |
C07C269/00 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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