发明名称 ANTIDIABETIC COMPOUNDS
摘要 The present invention provides novel peptidomimetics, of formula (I): A-Z<SUB>1</SUB>-Z<SUB>2</SUB>-Z<SUB>3</SUB>-Z<SUB>4</SUB>-Z<SUB>5</SUB>-Z<SUB>6</SUB>-Z<SUB>7</SUB>-Z<SUB>8</SUB>-Z<SUB>9</SUB>-Z<SUB>10</SUB>-Z<SUB>11</SUB>-B, which primarily act as glucose dependent insulin secretagogues. Furthermore, it was found that these peptidomimetics showed glucagon receptor antagonistic activity, along with the GLP-1 receptor agonistic activity.
申请公布号 WO2008062457(A3) 申请公布日期 2008.10.02
申请号 WO2007IN00457 申请日期 2007.09.28
申请人 CADILA HEALTHCARE LIMITED;BAHEKAR, RAJESH, H.;LOHRAY, BRAJ, BHUSHAN;LOHRAY, VIDYA, BHUSHAN;JAIN, MUKUL, R.;BANERJEE, KAUSHIK, M.;PATEL, PANKAJ, RAMANBHAI 发明人 BAHEKAR, RAJESH, H.;LOHRAY, BRAJ, BHUSHAN;LOHRAY, VIDYA, BHUSHAN;JAIN, MUKUL, R.;BANERJEE, KAUSHIK, M.;PATEL, PANKAJ, RAMANBHAI
分类号 C07K14/605 主分类号 C07K14/605
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