发明名称 Atropisomers of 3-substituted-4-arylquinolin-2-one derivatives for potassium channel regulation
摘要 The present disclosure provides pharmaceutical compositions comprising the atropisomers of 3-substituted-4-arylquinolin-2-one derivatives, as in fig 1, substituents of which are as defined in the specification, and methods for the treatment of conditions sensitive to potassium channel opening activity such as ischemia, stroke, convulsions, epilepsy, asthma, irritable bowel syndrome, migraine, traumatic brain injury, spinal cord injury, sexual dysfunction and urinary incontinence.
申请公布号 NZ541237(A) 申请公布日期 2008.09.26
申请号 NZ20030541237 申请日期 2003.12.18
申请人 BRISTOL-MYERS SQUIBB COMPANY 发明人 VRUDHULA, VIVEKANANDA M;GRIBKOFF, VALENTIN KALA;DASGUPTA, BIRESHWAR;BOISSARD, CHRISTOPHER G
分类号 C07D215/22;C07D215/227;(IPC1-7):A61K31/47;C07D215/16;C07D215/20 主分类号 C07D215/22
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